Based on our former development candidate BAY 38-1315, optimization efforts led to the discovery of a novel chemical class of orally active cholesteryl ester transfer protein (CETP) inhibitors. The chromanol derivative 19b is a highly potent CETP inhibitor with favorable pharmacokinetic properties s
✦ LIBER ✦
Dibenzodioxocinones—A new class of CETP inhibitors
✍ Scribed by David Brückner; Frank-Thorsten Hafner; Volkhart Li; Carsten Schmeck; Joachim Telser; Alexandros Vakalopoulos; Gabriele Wirtz
- Book ID
- 108073684
- Publisher
- Elsevier Science
- Year
- 2005
- Tongue
- English
- Weight
- 236 KB
- Volume
- 15
- Category
- Article
- ISSN
- 0960-894X
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