Diastereoselective Synthesis of Cyclopropyl Boronic Esters. -A simple and efficient protocol for the conversion of 1-alkynes to 2-alkylcyclopropanols is described. Thus, 1-alkyne-derived alkynyl boronic esters (I) are converted to chiral tartrates (IV) and then subjected to cyclopropanation providi
Diastereoselective synthesis of cyclopropyl melatonin analogues
✍ Scribed by Ann Hughes, Rachael; Tølløfsrud, Magnus; Bryant, Nathan; Kaboli, Massoud; Hennum, Martin; Bonge-Hansen, Tore
- Book ID
- 118164483
- Publisher
- Elsevier Science
- Year
- 2013
- Tongue
- French
- Weight
- 465 KB
- Volume
- 54
- Category
- Article
- ISSN
- 0040-4039
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