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Development of a Practical and Efficient Synthesis of SIPI-4884, a HMG CoA Reductase Inhibitor for the Treatment of Hypercholesterolemia

✍ Scribed by Hao, Qun; Pan, Jing; Li, Yongjia; Cai, Zhengyan; Zhou, Weicheng

Book ID
120397910
Publisher
American Chemical Society
Year
2013
Tongue
English
Weight
426 KB
Volume
17
Category
Article
ISSN
1083-6160

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On p. 1074, in Scheme 3, the correct formula of NK-104 should be as follows: 2) On p. 1077, line 16 should read as follows: (390 ml) was cooled to Γ€ 788, and 1.6m BuLi in hexane (374.4 g, 881 mmol) was added under 3) On p. 1078, line 15 should read as follows: As HPLC revealed the presence of mor