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Design, Synthesis, and Evaluation of Orally Active 4-(2,4-Difluoro-5-(methoxycarbamoyl)phenylamino)pyrrolo[2,1- f ][1,2,4]triazines as Dual Vascular Endothelial Growth Factor Receptor-2 and Fibroblast Growth Factor Receptor-1 Inhibitors

✍ Scribed by Borzilleri, Robert M.; Zheng, Xiaoping; Qian, Ligang; Ellis, Christopher; Cai, Zhen-wei; Wautlet, Barri S.; Mortillo, Steve; Jeyaseelan,, Robert; Kukral, Daniel W.; Fura, Aberra; Kamath, Amrita; Vyas, Viral; Tokarski, John S.; Barrish, Joel C.; Hunt, John T.; Lombardo, Louis J.; Fargnoli, Joseph; Bhide, Rajeev S.

Book ID: 118190595
Publisher: American Chemical Society
Year: 2005
Tongue: English
Weight: 459 KB
Volume: 48
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm0501275

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