Probes for narcotic receptor mediated ph
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Terrence R. Burke Jr.; Kenner C. Rice; Arthur E. Jacobson; William F. Simonds; W
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Article
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1984
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John Wiley and Sons
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French
β 381 KB
Tritiation of the delta-specific opioid alkylating ligand FIT, 3 and the mu-specific opioid alkylating ligand BIT, 2 to high specific activity is described. Both compounds were derived from dibrominated amino intermediates (4 and lo, respectively) which were tritiated with tritium gas over Pd/C befo