The percutaneous permeation characteristics of 6 potential prodrugs 2-7 in comparison with their parent drug mefenamic acid (1) in virro using excised human skin were studied. The results show that all potential prodrugs tested were at least 2.0 times as effective as mefenamic acid; compounds 2 and
โฆ LIBER โฆ
Cycloserine Fatty Acid Derivatives (VI) as Prodrugs: Synthesis, Degradation and in vitro Skin Permeability.
โ Scribed by Thorsteinn Thorsteinsson; Mar Masson; Tomi Jarvinen; Tapio Nevalainen; Thorsteinn Loftsson
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 27 KB
- Volume
- 33
- Category
- Article
- ISSN
- 0931-7597
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