## Abstract The synthesis of 6βphenylβatevirdine (17), a lipophilic derivative of the potent HIVβ1 reverse transcriptase inhibitor atevirdine (1), is described. The title compound was prepared from dithioacetale 2 __via__ keteneaminal 4 and the nitropyridine derivative 10. Unexpectedly, no anti HIV
ChemInform Abstract: Synthesis of 6-Phenyl-Atevirdine.
β Scribed by R. TROSCHUETZ; A. KARGER
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 30 KB
- Volume
- 29
- Category
- Article
- ISSN
- 0931-7597
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## Abstract The stereoselective synthesis of the title compound (VI) by reduction of (V) in the presence of CBSβoxazaborolidine is reported.
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