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ChemInform Abstract: Production Scale Synthesis of the Non-Nucleoside Reverse Transcriptase Inhibitor Atevirdine Mesylate (U-87,201E).

✍ Scribed by W. R. PERRAULT; K. P. SHEPHARD; L. A. LAPEAN; M. A. KROOK; P. J. DOBROWOLSKI; M. A. LYSTER; M. W. MCMILLAN; D. J. KNOECHEL; G. N. EVENSON; W. WATT; B. A. PEARLMAN

Publisher: John Wiley and Sons
Year: 2010
Weight: 30 KB
Volume: 28
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199738203

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✦ Synopsis

Production Scale Synthesis of the Non-Nucleoside Reverse Transcriptase Inhibitor Atevirdine Mesylate (U-87,201E). -The large-scale preparation of the title compound (VII) is used to produce multiton quantities of bulk drug used in phase II clinical trials. -(PERRAULT, W. R.; SHEP-

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