๐”– Bobbio Scriptorium
โœฆ   LIBER   โœฆ

ChemInform Abstract: Mild Method for the Synthesis of Thiazolines from Secondary and Tertiary Amides.

โœ Scribed by A. B. CHARETTE; P. CHUA

Publisher
John Wiley and Sons
Year
2010
Weight
31 KB
Volume
29
Category
Article
ISSN
0931-7597

No coin nor oath required. For personal study only.

โœฆ Synopsis

Mild Method for the Synthesis of Thiazolines from Secondary and Tertiary Amides.

-Base-promoted treatment of amides [cf. (I)] with triflic anhydride generates an iminium or imino triflate which reacts with an aminothiol directly to biologically interesting thiazolines. When optically pure cysteine ethyl ester (V) is used, no racemization is observed. -(CHARETTE,

๐Ÿ“œ SIMILAR VOLUMES

ChemInform Abstract: A New Mild Method f
ChemInform Abstract: A New Mild Method for the Cleavage of the Amide Bond: Conversion of Secondary and Tertiary Amides to Esters.
โœ A. B. CHARETTE; P. CHUA ๐Ÿ“‚ Article ๐Ÿ“… 2010 ๐Ÿ› John Wiley and Sons โš– 29 KB ๐Ÿ‘ 2 views

1998 amide formation, amide hydrolysis amide formation, amide hydrolysis O 0320 23 -069 A New Mild Method for the Cleavage of the Amide Bond: Conversion of Secondary and Tertiary Amides to Esters. -A variety of secondary and tertiary amides (I) (21 examples) is efficiently converted to the correspon