Synthesis and Receptor Binding Affinity of Conformationally Restricted Retinoic Acid Analogues. -Efforts to synthesize two conformationally restricted retinoids utilizing a cyclopropyl ring as bioisostere for the C9-C10 double bond are described. The attempted synthesis of the cisisomer leads mainl
โฆ LIBER โฆ
ChemInform Abstract: High Affinity Retinoic Acid Receptor Antagonists: Analogues of AGN 193109.
โ Scribed by Alan T. Johnson; Liming Wang; Samuel J. Gillett; Roshantha A. S. Chandraratna
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 30 KB
- Volume
- 30
- Category
- Article
- ISSN
- 0931-7597
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