Brominalion and bromoh)drox)lalion of oxazolidinones derived from cyclohexadienc have been studied in order to synlhctizc (\_+)-cpibatidine 18. Bromohydrox.wlation of compound 2 led to a polyfunctionalized halohydrin lla ~vhich could be furlher c.vclized to azabieyclol2.2. I Iheptan-2one 16 already
β¦ LIBER β¦
ChemInform Abstract: Expeditious Formal Synthesis of (.+-.)-Epibatidine Using Diastereoselective Bromohydroxylation of Aminocyclohexene Derivatives.
β Scribed by I. CABANAL-DUVILLARD; J.-F. BERRIEN; J. ROYER; H.-P. HUSSON
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 35 KB
- Volume
- 29
- Category
- Article
- ISSN
- 0931-7597
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