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ChemInform Abstract: Butyrophenone Analogues in the Carbazole Series: Synthesis and Determination of Affinities at D2 and 5-HT2A Receptors.

✍ Scribed by Christian F. Masaguer; Emilio Formoso; Enrique Ravina; Helena Tristan; M. Isabel Loza; Emilia Rivas; Jose Angel Fontenla

Publisher: John Wiley and Sons
Year: 2010
Weight: 34 KB
Volume: 30
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199917126

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✦ Synopsis

Butyrophenone Analogues in the Carbazole Series: Synthesis and Determination of Affinities at D 2 and 5-HT 2A Receptors.

-As a part of an ongoing research program on new CNS acting agents two approaches to compounds such as (VII) are presented. The most promising compound (VIIc), named QF 2004B, is chosen as candidate for further development. -

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