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ChemInform Abstract: A Short, Scaleable Synthesis of Both Enantiomers of 2-Benzoylsulfanyl-5-phthalimidopentanoic Acid from Ornithine.

✍ Scribed by K. E. HOLT; G. E. HUTTON; C. N. MORFITT; G. RUECROFT; S. J. C. TAYLOR; P. D. TIFFIN; N. TREMAYNE; M. WOODS

Publisher: John Wiley and Sons
Year: 2010
Weight: 28 KB
Volume: 29
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199808172

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✦ Synopsis

Starting from ornithine, an efficient scalable one-pot 3-step procedure for the synthesis of the enantiopure bromo acid (I) is reported. It can be easily converted to chiral benzoylsulfanyl derivative (III), an intermediate in the synthesis of MMP inhibitors. -(HOLT, K.

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