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ChemInform Abstract: 2-(3-Pyridyl)thiazolidine-4-carboxamide Derivatives. Part 2. Structure—Activity Relationships and Active Configuration of 2-(3-Pyridyl)thiazolidine-4-carboxamides as Platelet-Activating Factor Receptor Antagonists.

✍ Scribed by Takeshi Suzuki; ET AL. ET AL.

Publisher: John Wiley and Sons
Year: 2010
Weight: 32 KB
Volume: 30
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199912052

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✦ Synopsis

1999 condensation reactions condensation reactions O 0120 12 -052 2-(3-Pyridyl)thiazolidine-4-carboxamide Derivatives. Part 2. Structure-Activity Relationships and Active Configuration of 2-(3-Pyridyl)thiazolidine-4-carboxamides as Platelet-Activating Factor Receptor Antagonists. -In continuation of a recent work different types of heterocycles such as (V), (VIII), and (IX) are synthesized. None of the compounds is more active than YM264. The structure-activity relationships are discussed in detail [no yields are given for (V) and (VII)]. -(SUZUKI,

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