The fast and efficient carbon-14 labelling of the three potent H 3 antagonists NNC 38-1202, NNC 38-1384, and NNC 38-1401 is reported. The two-step synthetic sequence, which included a Knoevenagel reaction, provided the carbon-14-labelled compounds in 38-55% overall yield starting from [2-14 C]maloni
Carbon-14 labelling of 3-cyanoquinolines
✍ Scribed by John D. Olszewski; Dan M. Berger; Michael K. May
- Publisher
- John Wiley and Sons
- Year
- 2007
- Tongue
- French
- Weight
- 79 KB
- Volume
- 50
- Category
- Article
- ISSN
- 0022-2135
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