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Buspirone enhances benzodiazepine receptor binding in vivo

โœ Scribed by N.E. Goeders; Mary C. Ritz; M.J. Kuhar


Book ID
118955877
Publisher
Elsevier Science
Year
1988
Tongue
English
Weight
663 KB
Volume
27
Category
Article
ISSN
0028-3908

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Barbiturates have been reported to augment benzodiazepine receptor affinity in vitro, but their effects in vivo are uncertain. We determined benzodiazepine receptor binding in vivo by specific uptake of [3H]Ro15-1788 after barbiturate administration. Pentobarbital (30 mg/kg) increased receptor bindi