✦ LIBER ✦

Aspartate138 is required for the high-affinity ligand binding site but not for the low-affinity binding site of the β1-adrenoceptor

✍ Scribed by Shirin S. Joseph; William H. Colledge; Alberto J. Kaumann

Publisher: Springer-Verlag
Year: 2004
Tongue: English
Weight: 124 KB
Volume: 370
Category: Article
ISSN: 0028-1298
DOI: 10.1007/s00210-004-0962-1

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Trishomocubanes, a new class of selectiv

Trishomocubanes, a new class of selective and high affinity ligands for the sigma binding site

✍ Michael Kassiou; Vu H. Nguyen; Robert Knott; MacDonald J. Christie; Trevor W. Ha 📂 Article 📅 1996 🏛 Elsevier Science 🌐 English ⚖ 279 KB

The synthesis, receptor binding, and preliminary structural characterisation of trishomocubanes of types pentacyclo [5.4.0.02'6.03'l°.05'9]undecylamines and 4-azahexacyclo[5.4.1.0E'6.03'l°.05'9.08'll]dodecanes are described. These ligands demonstrated high selectivity and affinity for the sigma bind

Airway relaxant and anti-inflammatory pr

Airway relaxant and anti-inflammatory properties of a PDE4 inhibitor with low affinity for the high-affinity rolipram binding site

✍ Christian Martin; Rolf Göggel; Vittorio Dal Piaz; Claudia Vergelli; Maria Giovan 📂 Article 📅 2002 🏛 Springer-Verlag 🌐 English ⚖ 100 KB

(R)-3-(6-chloro-1-isopropylbenzimidazole

(R)-3-(6-chloro-1-isopropylbenzimidazole-4-carboxamido)quinuclidine: A high affinity ligand for the (R)-zacopride binding site

✍ L.A. Flippin; D.S. Carter; J. Berger; R.D. Clark; D.W. Bonhaus; E. Leung; R.M. E 📂 Article 📅 1996 🏛 Elsevier Science 🌐 English ⚖ 192 KB

The high-affinity binding site for tricy

The high-affinity binding site for tricyclic antidepressants resides in the outer vestibule of the serotonin transporter

✍ Subhodeep Sarker; René Weissensteiner; Ilka Steiner; Harald H Sitte; Gerhard F E 📂 Article 📅 2010 🏛 BioMed Central 🌐 English ⚖ 94 KB

Sarker et al.: The high-affinity binding site for tricyclic antidepressants resides in the outer vestibule of the serotonin transporter. BMC Pharmacology 2010 10(Suppl 1):A21.

Identification of high-affinity binding

Identification of high-affinity binding sites for the hepta-β-glucoside elicitor in membranes of the model legumesMedicago truncatulaandLotus japonicus

✍ François Côté; Kathy A. Roberts; Michael G. Hahn 📂 Article 📅 2000 🏛 Springer-Verlag 🌐 English ⚖ 220 KB

Super-high-affinity binding site for [3H

Super-high-affinity binding site for [3H]diazepam in the presence of Co2+, Ni2+, Cu2+, OR Zn2+

✍ S. Mizuno; N. Ogawa; A. Mori 📂 Article 📅 1982 🏛 Springer 🌐 English ⚖ 293 KB