A novel and simple solid phase synthesis ofunsymme~cal secondary amines was developed. The general methodology was applied to the synthesis of arylethanolamines and arylpropanolamines.
Aromatic annelation; application to the synthesis of unsymmetrical biphenyls.
β Scribed by Marcus A. Tius
- Publisher
- Elsevier Science
- Year
- 1981
- Tongue
- French
- Weight
- 227 KB
- Volume
- 22
- Category
- Article
- ISSN
- 0040-4039
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β¦ Synopsis
for the preparation of unsynunetrical biphenyls by elaboration of aromatic ketones is described.
The formation of cyclic products from acyclic precursors is an important objective in organic synthesis. --. (e) M. Guyot and C. kntzer, Bull. Sot Chim Fr -_. _* -.) 1843 (1967); m.p. 102'C.
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