✦ LIBER ✦

Argifin; efficient solid phase total synthesis and evalution of analogues of acyclic peptide

✍ Scribed by Toshiaki Sunazuka; Akihiro Sugawara; Kanami Iguchi; Tomoyasu Hirose; Kenichiro Nagai; Yoshihiko Noguchi; Yoshifumi Saito; Tsuyoshi Yamamoto; Hideaki Ui; Hiroaki Gouda; Kazuro Shiomi; Takeshi Watanabe; Satoshi Ōmura

Book ID: 108072615
Publisher: Elsevier Science
Year: 2009
Tongue: English
Weight: 672 KB
Volume: 17
Category: Article
ISSN: 0968-0896
DOI: 10.1016/j.bmc.2009.02.047

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Solid-phase synthesis of cyclic peptide

Solid-phase synthesis of cyclic peptide chitinase inhibitors: SAR of the argifin scaffold

✍ Dixon, Mark J. ;Nathubhai, Amit ;Andersen, Ole A. ;van Aalten, Daan M. F. ;Eggle 📂 Article 📅 2009 🏛 Royal Society of Chemistry 🌐 English ⚖ 522 KB

Solid-Phase Total Synthesis of Cyclospor

Solid-Phase Total Synthesis of Cyclosporine Analogues

✍ Soo Y. Ko; Roland M. Wenger 📂 Article 📅 1997 🏛 John Wiley and Sons 🌐 German ⚖ 645 KB

Syntheses of cyclosporine analogues are reported wherein the peptide couplings were achieved in solid phase. The Wang resin was used as the solid support, and the peptide couplings commenced with the residue 11 of the cyclosporine skeleton. The couplings proceeded in a stepwide manner up to the res

Solid phase synthesis of retro-inverso p

Solid phase synthesis of retro-inverso peptide analogues

✍ BONELLI, FABIO ;PESSI, ANTONELLO ;VERDINI, ANTONIO S. 📂 Article 📅 2009 🏛 Wiley (Blackwell Publishing) 🌐 English ⚖ 235 KB

Solid-Phase Total Synthesis of Oscillami

Solid-Phase Total Synthesis of Oscillamide Y and Analogues

✍ Marsh, Ian R.; Bradley, Mark; Teague, Simon J. 📂 Article 📅 1997 🏛 American Chemical Society 🌐 English ⚖ 180 KB

Total synthesis of a depsidomycin analog

Total synthesis of a depsidomycin analogue by convergent solid-phase peptide synthesis and macrolactonization strategy for antitubercular activity

✍ Venugopala K. Narayanaswamy; Fernando Albericio; Yacoob Mohamed Coovadia; Hendri 📂 Article 📅 2011 🏛 John Wiley and Sons 🌐 English ⚖ 177 KB

## Abstract Depsidomycin is a cyclic heptadepsi‐peptide isolated from the cultured broth of __Streptomyces lavendofoliae__ MI951‐62F2. It exhibits significant antimicrobial and immunosuppressive activity. The total synthesis of a depsidomycin analogue in which 1,2‐piperazine‐3‐carboxylic acid was s

Simple and efficient solid-phase synthes

Simple and efficient solid-phase synthesis of unprotected peptide aldehyde for peptide segment ligation

✍ Dominique Lelièvre; Hadjila Chabane; Agnès Delmas 📂 Article 📅 1998 🏛 Elsevier Science 🌐 French ⚖ 217 KB

We describe an efficient solid-phase synthesis of C-terminal peptide aldehyde. Making use of the stability of the PAM linker towards both acid and base conditions, a pentapeptide was synthesized starting from a PAM resin according to Fmoe/tBu chemistry. The side-chains were deprotected by TFA. The p