## Abstract A general and efficient procedure for the synthesis of __N__βarylβsubstituted 4βpiperidones was developed. The two step syntheses proceeded with an overall yield of 60%β83% using __L__βproline as the ligand for the Cu(I)βcatalyzed Ullmann amination followed by subsequent hydrolysis of r
β¦ LIBER β¦
An Improved Synthesis of N-Aryl and N-Heteroaryl Substituted Piperidones.
β Scribed by Uwe Schoen; Josef Messinger; M. Buckendahl; M. S. Prabhu; A. Konda
- Publisher
- John Wiley and Sons
- Year
- 2007
- Weight
- 30 KB
- Volume
- 38
- Category
- Article
- ISSN
- 0931-7597
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