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Agonist induction and conformational selection during activation of a G-protein-coupled receptor

✍ Scribed by László Hunyady; Georges Vauquelin; Patrick Vanderheyden

Book ID
117341006
Publisher
Elsevier Science
Year
2003
Tongue
English
Weight
403 KB
Volume
24
Category
Article
ISSN
0165-6147

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## Abstract Agonist‐selective signaling or ligand‐biased signaling of G protein‐coupled receptor (GPCR) has become the focus of an increasing number of laboratories. The principle of this concept is that agonist possesses different abilities to activate different signaling pathways. Current review