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Structural insights into agonist-induced activation of G-protein-coupled receptors

✍ Scribed by Xavier Deupi; Jörg Standfuss

Book ID
113883442
Publisher
Elsevier Science
Year
2011
Tongue
English
Weight
1004 KB
Volume
21
Category
Article
ISSN
0959-440X

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## Abstract It has been recently established that G‐protein‐coupled receptors (GPCRs) can be constitutively active, i.e., they can be active in the absence of an agonist. This activity can be inhibited by so‐called inverse agonists. For a number of GPCRs, such inverse agonists have been developed a