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A regio- and stereoselective synthesis of substituted piperidones

✍ Scribed by Philippe Bayard; Léon Ghosez

Publisher
Elsevier Science
Year
1988
Tongue
French
Weight
177 KB
Volume
29
Category
Article
ISSN
0040-4039

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✦ Synopsis

The new activated 2-aza-1,3-dienes 1 are readily prepared by acylation of N-tri-methylsilylimines 3. They react with electrophilic olefins to yield substituted piperidones 4 _ and 6 with high diastereoselectivity.

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## Abstract ChemInform is a weekly Abstracting Service, delivering concise information at a glance that was extracted from about 200 leading journals. To access a ChemInform Abstract, please click on HTML or PDF.