A Novel Solid-Phase Approach to 2,4-Diaminothiazoles
✍ Scribed by Baer, Roman; Masquelin, Thierry
- Book ID
- 118048011
- Publisher
- American Chemical Society
- Year
- 2001
- Tongue
- English
- Weight
- 45 KB
- Volume
- 3
- Category
- Article
- ISSN
- 1520-4766
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The synthesis of Agel 416, an acylpolyamine derived from the spider Agenolopsis aperta, has been achieved on solid support. Stepwise synthesis of the polyamine chain was accomplished using N-protected amino alcohols and the Fukuyama±Mitsunobu reaction.