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A convenient one-pot procedure for the synthesis of 2-aryl quinazolines using active MnO2 as oxidant

✍ Scribed by Yi-Yuan Peng; Yuyun Zeng; Ganyinsheng Qiu; Lisheng Cai; Victor W. Pike

Publisher
Journal of Heterocyclic Chemistry
Year
2010
Tongue
English
Weight
106 KB
Volume
47
Category
Article
ISSN
0022-152X

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✦ Synopsis

Abstract

magnified image A variety of 2‐aryl quinazolines were synthesized from the condensation of 2‐aminobenzylamines and aryl aldehydes to form 2‐aryl‐1,2,3,4‐tetrahydroquinazolines and subsequent oxidation of the intermediates with MnO~2~. J. Heterocyclic Chem., (2010).

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