A Convenient Large-Scale Synthesis of Ethyl (2-Cyanoimino-5,6dichloro-1,2,3,4-tetrahydroquinazoline-3-yl)acetate. -A practical industrial scale synthesis of the title compound (III), a key intermediate in the synthesis of the drug anagrelide, starting from glycinate (I) is accomplished.
✦ LIBER ✦
A Convenient, Large-Scale Synthesis of 4′-Carboxamido N-Boc-2′,6′-dimethyl-L-phenylalanines.
✍ Scribed by Chaozhong Cai; Henry J. Breslin; Wei He
- Publisher
- John Wiley and Sons
- Year
- 2005
- Weight
- 20 KB
- Volume
- 36
- Category
- Article
- ISSN
- 0931-7597
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