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A comparison of acid labile linkage agents for the synthesis of peptide C-terminal amides

✍ Scribed by Michael S. Bernatowicz; Scott B. Daniels; Hubert Köster

Publisher
Elsevier Science
Year
1989
Tongue
French
Weight
261 KB
Volume
30
Category
Article
ISSN
0040-4039

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✦ Synopsis

linkage agents useful for the so1id phase peptic synthesis of C-terminal d&s were evaluated for their relative lability toward trifluoroacetic acid. The twomst reactive linkage agents StUdied*re cved in the synthesis of two different peptide amides by the Na-9-fluoreny~~Yloxycarbony1 protecting group strategy.

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