A simple three-step method for the solution-phase combinatorial synthesis of 2,6,9trisubstituted purines from 2,6-dichloropmine is described. The synthesis exploits the use of resin capture to remove excess reagent used in the f'mal step.
✦ LIBER ✦
8-Bromination of 2,6,9-trisubstituted purines with pyridinium tribromide
✍ Scribed by Bliman, David; Pettersson, Mariell; Bood, Mattias; Grøtli, Morten
- Book ID
- 121673637
- Publisher
- Elsevier Science
- Year
- 2014
- Tongue
- French
- Weight
- 434 KB
- Volume
- 55
- Category
- Article
- ISSN
- 0040-4039
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## Abstract For Abstract see ChemInform Abstract in Full Text.
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