✦ LIBER ✦

5‘- O -Tritylinosine and Analogues as Allosteric Inhibitors of Human Thymidine Phosphorylase

✍ Scribed by Casanova, Elena; Hernández, Ana-Isabel; Priego, Eva-María; Liekens, Sandra; Camarasa, María-José; Balzarini, Jan; Pérez-Pérez, María-Jesús

Book ID: 126799252
Publisher: American Chemical Society
Year: 2006
Tongue: English
Weight: 145 KB
Volume: 49
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm0605379

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

6-SUBSTITUTED 5-FLUOROURACIL DERIVATIVES

6-SUBSTITUTED 5-FLUOROURACIL DERIVATIVES AS TRANSITION STATE ANALOGUE INHIBITORS OF THYMIDINE PHOSPHORYLASE

✍ Kalman, Thomas I.; Lai, Li 📂 Article 📅 2005 🏛 Taylor and Francis Group 🌐 English ⚖ 264 KB

Discovery of 5-Substituted-6-chlorouraci

Discovery of 5-Substituted-6-chlorouracils as Efficient Inhibitors of Human Thymidine Phosphorylase

✍ Nencka, Radim; Votruba, Ivan; Hřebabecký, Hubert; Jansa, Petr; Tloušt'ová, Eva; 📂 Article 📅 2007 🏛 American Chemical Society 🌐 English ⚖ 258 KB

Aminoimidazolylmethyluracil Analogues as

Aminoimidazolylmethyluracil Analogues as Potent Inhibitors of Thymidine Phosphorylase and Their Bioreductive Nitroimidazolyl Prodrugs

✍ Reigan, Philip; Edwards, Philip N.; Gbaj, Abdul; Cole, Christian; Barry, Simon T 📂 Article 📅 2005 🏛 American Chemical Society 🌐 English ⚖ 307 KB

ChemInform Abstract: Synthesis of 5-Halo

ChemInform Abstract: Synthesis of 5-Halogeno-6-amino-2′-deoxyuridines and Their Analogues as Potential Inhibitors of Thymidine Phosphorylase.

✍ Bai-Chuan Pan; Zhi-Hao Chen; Edward Chu; Ming-Yu Wang Chu; Shih-Hsi Chu 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 31 KB 👁 2 views

Synthesis and Evaluation of Thymidine-5′

Synthesis and Evaluation of Thymidine-5′-O-monophosphate Analogues as Inhibitors of Mycobacterium tuberculosis Thymidylate Kinase.

✍ Veerle Vanheusden; Helene Munier-Lehmann; Sylvie Pochet; Piet Herdewijn; Serge V 📂 Article 📅 2003 🏛 John Wiley and Sons ⚖ 78 KB 👁 2 views

Identification of aspartic acid-203 in h

Identification of aspartic acid-203 in human thymidine phosphorylase as an important residue for both catalysis and non-competitive inhibition by the small molecule “crystallization chaperone” 5′-O-tritylinosine (KIN59)

✍ A. Bronckaers; L. Aguado; A. Negri; M.-J. Camarasa; J. Balzarini; M.-J. Pérez-Pé 📂 Article 📅 2009 🏛 Elsevier Science 🌐 English ⚖ 766 KB