4-Azido[3,5-[3H]]phenacylbromide, a versatile bifunctional reagent for photoaffinity radiolabeling. Synthesis of prostaglandin 4-azido[3,5-[3H]]phenacyl esters
β Scribed by Smith, Bradley D.; Nakanishi, Koji; Watanabe, Kikuko; Ito, Seiji
- Book ID
- 121306942
- Publisher
- American Chemical Society
- Year
- 1990
- Tongue
- English
- Weight
- 259 KB
- Volume
- 1
- Category
- Article
- ISSN
- 1043-1802
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An efficient preparation of the title compound la starting from propargyl alcohol and proceeding via deuterated monomethyl adipate (&) is described. As demonstrated by t h e first total synthesis of deuterated w-carboxy-thromboxane B2 (&I, may serve as a versatile starting compound for t h e synthes
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