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2-Heterocyclic indole-3-sulfones as inhibitors of HIV-1 reverse transcriptase

✍ Scribed by Steven D. Young; Muriel C. Amblard; Susan F. Britcher; Vanessa E. Grey; Lee O. Tran; William C. Lumma; Joel R. Huff; William A. Schleif; Emilio E. Emini; Julie A. O'Brien; Douglas J. Pettibone


Book ID
103982849
Publisher
Elsevier Science
Year
1995
Tongue
English
Weight
265 KB
Volume
5
Category
Article
ISSN
0960-894X

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Pyridazines 92. Synthesis of dialkyldipy
✍ Gottfried Heinisch; Barbara Matuszczak; Elisabeth Spielmann; Myriam Witvrouw; Ch πŸ“‚ Article πŸ“… 2001 πŸ› Journal of Heterocyclic Chemistry 🌐 English βš– 71 KB

## Abstract Two methods for the preparation of dialkylsubstituted dipyridazino[4,3‐__b__:3β€²,4′‐__e__][1,4]diazepinones and dipyridazino[3,4‐__b__:3β€²,4′‐__e__][1,4]diazepinones are reported. The new compounds were evaluated for their inhibitory effects against the replication of human immunodeficien