The development of a novel series of non
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P. Boden; J.M. Eden; J. Hodgson; D.C. Horwell; M.C. Pritchard; J. Raphy; N. Suma
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Article
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1995
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Elsevier Science
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English
β 222 KB
In this paper we describe the transformation of a series of modified dipeptide NK 3 receptor selective ligands, previously developed from a hit identified from the screening of a dipeptide chemical library, into non-peptide, nanomolar affinity NK 3 receptor selective antagonists eg. PD160946 and PD1