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Transformations of Methyl 2-[(E)-2-(Dimethylamino)-1-(methoxycarbonyl)ethenyl]-1-methyl-1H-indole-3-carboxylate

✍ Scribed by David Bevk; Uroš Grošelj; Anton Meden; Jurij Svete; Branko Stanovnik

Publisher: John Wiley and Sons
Year: 2006
Tongue: German
Weight: 121 KB
Volume: 89
Category: Article
ISSN: 0018-019X
DOI: 10.1002/hlca.200690248

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✦ Synopsis

A simple and efficient synthesis of novel 2-heteroaryl-substituted 1H-indole-2-carboxylates and gcarbolines, compounds 1 -3, from methyl 2-(2-methoxy-2-oxoethyl)-1-methyl-1H-indole-3-carboxylate (4) by the enaminone methodology is presented.

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