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Transformations of methyl 2-(2,2-disubstituted-ethenyl)amino-3-dimethylaminopropenoates. The synthesis of methyl 1-heteroaryl-1H-imidazole-4-carboxylates

✍ Scribed by Lovro Selič; Branko Stanovnik

Publisher
Journal of Heterocyclic Chemistry
Year
1998
Tongue
English
Weight
182 KB
Volume
35
Category
Article
ISSN
0022-152X

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✦ Synopsis

Abstract

Transformations of intermediates 4, prepared from methyl 2‐(2,2‐disubstituted‐ethenyl)amino‐3‐dimethylaminopropenoates 2 and sterically hindered heteroarylamines 3, into methyl 1‐heteroaryl‐1__H__‐imidazole‐4‐carboxylates 7 are described.

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