Total synthesis of the marine pyridoacri
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Laurent Legentil; Jean Bastide; Evelyne Delfourne
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Article
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2003
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Elsevier Science
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French
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The synthesis of the marine alkaloid sebastianine A and of a regioisomer has been accomplished via hetero-Diels-Alder reaction of indole-4,7-dione or N-tosylindole-4,7-dione with trifluoroacetamidocinnamaldehyde dimethylhydrazone, and subsequent cyclisation in alkaline conditions.