Total syntheses of 6- and 7-azaindole derived GnRH antagonists
โ Scribed by Feroze Ujjainwalla; Thomas F Walsh
- Book ID
- 104231378
- Publisher
- Elsevier Science
- Year
- 2001
- Tongue
- French
- Weight
- 88 KB
- Volume
- 42
- Category
- Article
- ISSN
- 0040-4039
No coin nor oath required. For personal study only.
โฆ Synopsis
The palladium(0)-catalyzed heteroannulation of a triethylsilyl alkyne and an ortho-aminoiodopyridine derivative is used as the key step in a highly convergent route to 6-and 7-azaindoles of biological interest.
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