✦ LIBER ✦

The screening of enzyme-targeted drugs

✍ Scribed by C. L. Tsou

Book ID: 101710445
Publisher: John Wiley and Sons
Year: 1987
Tongue: English
Weight: 262 KB
Volume: 6
Category: Article
ISSN: 0265-9247
DOI: 10.1002/bies.950060511

No coin nor oath required. For personal study only.

✦ Synopsis

In this article C . L. Tsou, of the Institute of Biophysics, Beijing, criticizes the use of the expression I,,, the inhibitor concentration to produce 50% inhibition of a particular enzyme as a 'most unfortunate' parameter, when screening enzyme inhibitors designed as drugs. Comments on Dr Tsou's point of view will be welcomed from readers.

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