✦ LIBER ✦

The enantiomers of epiboxidine and of two related analogs: Synthesis and estimation of their binding affinity at α4β2 and α7 neuronal nicotinic acetylcholine receptors

✍ Scribed by Clelia Dallanoce; Carlo Matera; Marco De Amici; Luca Rizzi; Luca Pucci; Cecilia Gotti; Francesco Clementi; Carlo De Micheli

Book ID: 112049482
Publisher: John Wiley and Sons
Year: 2012
Tongue: English
Weight: 251 KB
Volume: 24
Category: Article
ISSN: 0899-0042
DOI: 10.1002/chir.22052

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Synthesis and binding affinity at α4β2 a

Synthesis and binding affinity at α4β2 and α7 nicotinic acetylcholine receptors of new analogs of epibatidine and epiboxidine containing the 7-azabicyclo[2.2.1]hept-2-ene ring system

✍ Clelia Dallanoce; Carlo Matera; Luca Pucci; Cecilia Gotti; Francesco Clementi; M 📂 Article 📅 2012 🏛 Elsevier Science 🌐 English ⚖ 617 KB

Synthesis of Epibatidine-Related Δ2-Isox

Synthesis of Epibatidine-Related Δ2-Isoxazoline Derivatives and Evaluation of Their Binding Affinity at Neuronal Nicotinic Acetylcholine Receptors

✍ Clelia Dallanoce; Paola Bazza; Giovanni Grazioso; Marco De Amici; Cecilia Gotti; 📂 Article 📅 2006 🏛 John Wiley and Sons 🌐 English ⚖ 193 KB

New Analogues of Epiboxidine Incorporati

New Analogues of Epiboxidine Incorporating the 4,5-Dihydroisoxazole Nucleus: Synthesis, Binding Affinity at Neuronal Nicotinic Acetylcholine Receptors, and Molecular Modeling Investigations

✍ Clelia Dallanoce; Pietro Magrone; Paola Bazza; Giovanni Grazioso; Luca Rizzi; Lo 📂 Article 📅 2009 🏛 John Wiley and Sons 🌐 English ⚖ 454 KB 👁 1 views

## Abstract magnified image A group of novel 4,5‐dihydro‐3‐methylisoxazolyl derivatives, structurally related to epiboxidine (=(1__R__,4__S__,6__S__)‐6‐(3‐methylisoxazol‐5‐yl)‐7‐azabicyclo[2.2.1]heptane), was prepared __via__ 1,3‐dipolar cycloaddition of acetonitrile oxide to different olefins. Ta

Low-affinity Ca2+ and Ba2+ binding sites

Low-affinity Ca2+ and Ba2+ binding sites in the pore of α7 nicotinic acetylcholine receptors

✍ L.K. Lyford; J.W. Lee; R.L. Rosenberg 📂 Article 📅 2002 🏛 Elsevier Science 🌐 English ⚖ 460 KB

Structural differences determine the rel

Structural differences determine the relative selectivity of nicotinic compounds for native α4β2*-, α6β2*-, α3β4*- and α7-nicotine acetylcholine receptors

✍ Sharon R. Grady; Ryan M. Drenan; Scott R. Breining; Daniel Yohannes; Charles R. 📂 Article 📅 2010 🏛 Elsevier Science 🌐 English ⚖ 620 KB

Synthesis and binding affinities of 5-(3

Synthesis and binding affinities of 5-(3-pyridinyl)- and 5-(3-quinolinyl)-4-azahomoadamantanes to α7 nicotinic acetylcholine receptors

✍ Dimitris Tataridis; Antonios Kolocouris; George Fytas; Nicolas Kolocouris; Georg 📂 Article 📅 2002 🏛 Elsevier Science 🌐 English ⚖ 167 KB