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The design and synthesis of 5- and 6-isoxazolylbenzimidazoles as selective inhibitors of the BET bromodomains

✍ Scribed by Hay, Duncan ;Fedorov, Oleg ;Filippakopoulos, Panagis ;Martin, Sarah ;Philpott, Martin ;Picaud, Sarah ;Hewings, David S. ;Uttakar, Sagar ;Heightman, Tom D. ;Conway, Stuart J. ;Knapp, Stefan ;Brennan, Paul E.

Book ID: 120553662
Publisher: The Royal Society of Chemistry
Year: 2013
Tongue: English
Weight: 274 KB
Volume: 4
Category: Article
ISSN: 2040-2503
DOI: 10.1039/C2MD20189E

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