The Discovery of I-BET726 (GSK1324726A), a Potent Tetrahydroquinoline ApoA1 Up-Regulator and Selective BET Bromodomain Inhibitor

✍ Scribed by Gosmini, Romain; Nguyen, Van Loc; Toum, Jérôme; Simon, Christophe; Brusq, Jean-Marie G.; Krysa, Gael; Mirguet, Olivier; Riou-Eymard, Alizon M.; Boursier, Eric V.; Trottet, Lionel; Bamborough, Paul; Clark, Hugh; Chung, Chun-wa; Cutler, Leanne; Demont, Emmanuel H.; Kaur, Rejbinder; Lewis, Antonia J.; Schilling, Mark B.; Soden, Peter E.; Taylor, Simon; Walker, Ann L.; Walker, Matthew D.; Prinjha, Rab K.; Nicodème, Edwige

• Book ID: 126785549
• Publisher: American Chemical Society
• Year: 2014
• Tongue: English
• Weight: 963 KB
• Volume: 57
• Category: Article
• ISSN: 0022-2623
• DOI: 10.1021/jm5010539