A series of 5'-halogenated resiniferatoxin analogs have been investigated in order to examine the effect of halogenation in the A-region on their binding and the functional pattern of agonism/antagonism for rat TRPV1 heterologously expressed in Chinese hamster ovary cells. Halogenation at the 5-posi
✦ LIBER ✦
The carbonate analogues of 5′-halogenated resiniferatoxin as TRPV1 ligands
✍ Scribed by Lim, Kwang Su; Lee, Hobin; Kim, Sung Eun; Ha, Tae-Hwan; Ann, Jihyae; Son, Karam; Choi, Sun; Sun, Wei; Pearce, Larry V.; DeAndrea-Lazarus, Ian A.; Blumberg, Peter M.; Lee, Jeewoo
- Book ID
- 123385802
- Publisher
- Elsevier Science
- Year
- 2013
- Tongue
- French
- Weight
- 833 KB
- Volume
- 68
- Category
- Article
- ISSN
- 0223-5234
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