✦ LIBER ✦

Target Profiling of a Small Library of Phosphodiesterase 5 (PDE5) Inhibitors using Chemical Proteomics

✍ Scribed by Dr. Reinout Raijmakers; Dr. Poupak Dadvar; Dr. Sarah Pelletier; Dr. Joost Gouw; Dr. Klaus Rumpel; Prof. Dr. Albert J. R. Heck

Book ID: 102804341
Publisher: John Wiley and Sons
Year: 2010
Tongue: English
Weight: 588 KB
Volume: 5
Category: Article
ISSN: 1860-7179
DOI: 10.1002/cmdc.201000303

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Effects of a phosphodiesterase-5 (PDE5)

Effects of a phosphodiesterase-5 (PDE5) inhibitor on endothelium-dependent relaxation of myometrial small arteries

✍ Mark Wareing; Jenny E Myers; Maureen O'Hara; Louise C Kenny; Averil Y Warren; Mi 📂 Article 📅 2004 🏛 Elsevier Science 🌐 English ⚖ 230 KB

Utilization of Halogen Bond in Lead Opti

Utilization of Halogen Bond in Lead Optimization: A Case Study of Rational Design of Potent Phosphodiesterase Type 5 (PDE5) Inhibitors

✍ Xu, Zhijian; Liu, Zheng; Chen, Tong; Chen, TianTian; Wang, Zhen; Tian, Guanghui; 📂 Article 📅 2011 🏛 American Chemical Society 🌐 English ⚖ 789 KB

1253 A SYSTEMATIC REVIEW AND META-ANALYS

1253 A SYSTEMATIC REVIEW AND META-ANALYSIS OF THE USE OF PHOSPHODIESTERASE TYPE 5 INHIBITORS (PDE5-IS) FOR LOWER URINARY TRACT SYMPTOMS (LUTS) SECONDARY TO BENIGN PROSTATIC HYPERPLASIA (BPH)

✍ Gacci, Mauro; Corona, Giovanni; Salvi, Matteo; Vignozzi, Linda; McVary, Kevin T. 📂 Article 📅 2012 🏛 Lippincott Williams and Wilkins 🌐 English ⚖ 112 KB

Discovery of Potent Chromen-4-one Inhibi

Discovery of Potent Chromen-4-one Inhibitors of the DNA-Dependent Protein Kinase (DNA-PK) Using a Small-Molecule Library Approach

✍ Hardcastle, Ian R.; Cockcroft, Xiaoling; Curtin, Nicola J.; El-Murr, Marine Desa 📂 Article 📅 2005 🏛 American Chemical Society 🌐 English ⚖ 429 KB

Discovery of Highly Potent and Selective

Discovery of Highly Potent and Selective Small Molecule ADAMTS-5 Inhibitors That Inhibit Human Cartilage Degradation via Encoded Library Technology (ELT)

✍ Deng, Hongfeng; O’Keefe, Heather; Davie, Christopher P.; Lind, Kenneth E.; Achar 📂 Article 📅 2012 🏛 American Chemical Society 🌐 English ⚖ 689 KB

Correction to Mitogen-Activated Protein

Correction to Mitogen-Activated Protein Kinase-Activated Protein Kinase 2 (MAPKAP-K2) as an Antiinflammatory Target: Discovery and in Vivo Activity of Selective Pyrazolo[1,5- a ]pyrimidine Inhibitors Using a Focused Library and Structure-Based Optimization Approach

✍ Kosugi, Tomomi; Mitchell, Dale R.; Fujino, Aiko; Imai, Minoru; Kambe, Mika; Koba 📂 Article 📅 2012 🏛 American Chemical Society 🌐 English ⚖ 174 KB