Tandem Heck—Suzuki—Miyaura Reaction: Application to the Synthesis of Constrained Analogues of Combretastatin A-4.
✍ Scribed by Martin Arthuis; Renee Pontikis; Jean-Claude Florent
- Book ID
- 102012600
- Publisher
- John Wiley and Sons
- Year
- 2007
- Weight
- 23 KB
- Volume
- 38
- Category
- Article
- ISSN
- 0931-7597
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Heck reactions of unsaturated amino acid building blocks are described which allow access to homo-and bishomophenylalanine derivatives and to g,d-unsaturated amino acids. Preliminary synthetic studies utilising this chemistry for the preparation of pyrrololine and deoxypyrrololine analogues are also
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