Synthetic studies on teleocidin I. Regioselective introduction of 4-amino and 7-acyl groups on indole derivative

Synthetic studies on teleocidin II. Synt

Synthetic studies on teleocidin II. Synthesis of indole derivatives containing the same substituent to teleocidin bat 6- and 7-positions of indole nucleus.

✍ Shin-ichi Nakatsuka; Toshiya Masuda; Toshio Goto 📂 Article 📅 1986 🏛 Elsevier Science 🌐 French ⚖ 240 KB

The same substituent to teleocidin B at 6-and 7-positions of indole nucleus was introduced via intramolecular cyclization and oxidative cleavage of C-N bond at l-position starting from simple indole. Teleocidin B (k) 2) 1s one of the most interesting natural products because of its potent biological