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Synthesis, Structure−Activity Relationships, and Biological Profiles of a Quinazolinone Class of Histamine H 3 Receptor Inverse Agonists

✍ Scribed by Nagase, Tsuyoshi; Mizutani, Takashi; Ishikawa, Shiho; Sekino, Etsuko; Sasaki, Takahide; Fujimura, Takashi; Ito, Sayaka; Mitobe, Yuko; Miyamoto, Yasuhisa; Yoshimoto, Ryo; Tanaka, Takeshi; Ishihara, Akane; Takenaga, Norihiro; Tokita, Shigeru; Fukami, Takehiro; Sato, Nagaaki

Book ID: 125931294
Publisher: American Chemical Society
Year: 2008
Tongue: English
Weight: 170 KB
Volume: 51
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm8003834

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## Abstract **H**~**3**~**R inverse agonists** based on an aminopropoxy‐phenyloxazoline framework constitute highly valuable druglike lead compounds that display efficacy in a mouse model of recognition memory.magnified image