✦ LIBER ✦

Discovery of a New Class of Non-imidazole Oxazoline-Based Histamine H3 Receptor (H3R) Inverse Agonists

✍ Scribed by Sylvain Célanire; Maikel Wijtmans; Bernard Christophe; Philippe Collart; Iwan de Esch; Donald Dassesse; Christel Delaunoy; Frédéric Denonne; Véronique Durieu; Edith Gelens; Michel Gillard; Bénédicte Lallemand; Yves Lamberty; Florence Lebon; Jean-Marie Nicolas; Luc Quéré; Erwin Snip; Alain Vanbellinghen; Nathalie Van houtvin; Valérie Verbois; Henk Timmerman; Patrice Talaga; Rob Leurs; Laurent Provins

Publisher: John Wiley and Sons
Year: 2009
Tongue: English
Weight: 428 KB
Volume: 4
Category: Article
ISSN: 1860-7179
DOI: 10.1002/cmdc.200900055

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✦ Synopsis

Abstract

H~3~R inverse agonists based on an aminopropoxy‐phenyloxazoline framework constitute highly valuable druglike lead compounds that display efficacy in a mouse model of recognition memory.magnified image

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