✦ LIBER ✦

Synthesis of (β-methyl3H-6β-iodopenicillanic acid

✍ Scribed by Fabien De Meester; Jean-Marie Frère; Jean-Louis Piette; Hubert Vanderhaeghe

Publisher: John Wiley and Sons
Year: 1985
Tongue: French
Weight: 428 KB
Volume: 22
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580220502

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✦ Synopsis

A rapid and easy synthesis of tritium-labelled 8-iodopenicillanate, an efficient inactivator of serine B-lactamase, is described. This method involves only three reaction steps after the introduction of the label in the molecule with an overall yield of 16 % .

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