## Abstract [D~2~](1__R__)‐3‐methyl‐1‐[[(2S)‐1‐oxo‐3‐phenyl‐2‐[(pyrazinylcarbonyl)amino]propyl]‐amino]butyl] boronic acid ([D~2~]bortezomib), a proteasome inhibitor, was synthesized in 11 steps from __iso__butyryl chloride. Key steps in the synthesis included formation of the __iso__butyryl boronic
Synthesis of two labeled forms of proteasome inhibitor MLN273
✍ Scribed by Mihaela Plesescu; Yuexian Li; Shimoga R. Prakash
- Publisher
- John Wiley and Sons
- Year
- 2007
- Tongue
- French
- Weight
- 88 KB
- Volume
- 50
- Category
- Article
- ISSN
- 0022-2135
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