✦ LIBER ✦

Synthesis of tritium labeled 1-amidino-3-(P-nitro-phenyl)urea: A potential antimalarial agent

✍ Scribed by Theodore S. T. Wang; Rashid A. Fawwaz; Ronald L. van Heertum

Publisher: John Wiley and Sons
Year: 1993
Tongue: French
Weight: 219 KB
Volume: 33
Category: Article
ISSN: 0022-2135
DOI: 10.1002/jlcr.2580330904

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✦ Synopsis

Abstract

Five steps were required to synthesize the title compound. This involved a catalytic exchange reaction, nitration, hydrolysis, and condensation. The overall radiochemical yield was 28.87% and the specific activity was 12.4 mCi/mmol, with a radiochemical purity of more than 95.7%.

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