✦ LIBER ✦

Synthesis of Stereodefined 3,4-Disubstituted Piperidines through Rearrangement of 2-(2-Bromo-1,1-dimethylethyl)azetidines

✍ Scribed by D’hooghe, Matthias; De Kimpe, Norbert; Mollet, Karen; Broeckx, Leen

Book ID: 118145944
Publisher: Japan Institute of Heterocyclic Chemistry
Year: 2012
Tongue: English
Weight: 767 KB
Volume: 84
Category: Article
ISSN: 0385-5414
DOI: 10.3987/com-11-s(p)3

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

ChemInform Abstract: Synthesis of Stereo

ChemInform Abstract: Synthesis of Stereodefined 3,4-Disubstituted Piperidines Through Rearrangement of 2-(2-Bromo-1,2-dimethylethyl)azetidines.

✍ Karen Mollet; Leen Broeckx; Matthias D'hooghe; Norbert de Kimpe 📂 Article 📅 2012 🏛 John Wiley and Sons ⚖ 39 KB

Synthesis of piperidin-4-ones starting f

Synthesis of piperidin-4-ones starting from 2-(2-bromo-1,1-dimethylethyl)azetidines and 2-(2-mesyloxyethyl)azetidines through a ring expansion–oxidation protocol

✍ Mollet, Karen; D'hooghe, Matthias; Broeckx, Leen; Danneels, Barbara; Desmet, Tom 📂 Article 📅 2013 🏛 Elsevier Science 🌐 French ⚖ 229 KB

ChemInform Abstract: Stereoselective Syn

ChemInform Abstract: Stereoselective Synthesis of cis-3,4-Disubstituted Piperidines Through Ring Transformation of 2-(2-Mesyloxyethyl)azetidines.

✍ Karen Mollet; Saron Catak; Michel Waroquier; Veronique Van Speybroeck; Matthias 📂 Article 📅 2012 🏛 John Wiley and Sons ⚖ 38 KB 👁 2 views

Facile Stereoselective Synthesis of 1,3-

Facile Stereoselective Synthesis of 1,3-Disubstituted-4-trichloromethyl Azetidin-2-ones.

✍ V. V. Govande; A. R. A. S. Deshmukh 📂 Article 📅 2004 🏛 John Wiley and Sons ⚖ 22 KB 👁 2 views

1,4-Dehydrobromination of 1-bromo-1,2,3-

1,4-Dehydrobromination of 1-bromo-1,2,3-butatrienes: an efficient synthesis of 1,4-disubstituted 1,3-diynes

✍ Ziegler, Carl B.; Harris, Sonja M.; Baldwin, J. E. 📂 Article 📅 1987 🏛 American Chemical Society 🌐 English ⚖ 526 KB

Two-Step Synthesis of 1,3-Disubstituted

Two-Step Synthesis of 1,3-Disubstituted 3,4-Dihydro-4-thioxoquinazolin-2(1H)-ones from 1-Bromo-2-fluorobenzenes

✍ Kazuhiro Kobayashi; Toshihide Komatsu; Yuki Yokoi; Hisatoshi Konishi 📂 Article 📅 2011 🏛 John Wiley and Sons 🌐 German ⚖ 141 KB 👁 1 views

## Abstract An efficient synthesis of 3‐alkyl‐3,4‐dihydro‐4‐thioxobenzoquinazolin‐2(1__H__)‐ones **3** has been accomplished in two steps and in satisfactory yields from 1‐bromo‐2‐fluorobenzenes **1**. Thus, the reaction of 1‐fluoro‐2‐lithiobenzenes, generated by the Br/Li exchange between **1** an